Synthesis and Characterizations of (2Z)-ethyl-2-(Aryl)-3,5,8,8a-tetrahydro-5-(4-methoxyphenyl)-7-methyl-3-oxo-2H-oxazolo[3,2-a]pyrimidine-6-carboxylate as Biological Active Agents

Authors

  • J. S. Makwana  Department of Chemistry, M. G. Science institute, Navarangpura, Ahmedabad, Gujarat, India
  • Dr. B. B. Baldaniya  Department of Chemistry, M. G. Science institute, Navarangpura, Ahmedabad, Gujarat, India

Keywords:

Oxazolo Pyrimidine, Antibacterial activity, antifungal activities, Biginelli reaction.

Abstract

Pyrimidine plays a significant role among other heterocycles. Pyrimidine nucleus was synthesized by Biginelli reaction. The purpose of this study was to synthesize several oxazolo derivative compounds (1-13) and evaluate them for their antibacterial activity. The structures of all title compounds have been confirmed on the basis of their analytical, IR spectral data. The title compounds have been tested for antibacterial and antifungal activities against different strains of bacteria.

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International Journal of Scientific Research in Science and Technology

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Published

2017-04-30

Issue

Volume 3, Issue 3, March-April-2017

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Research Articles

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How to Cite

[1]
J. S. Makwana, Dr. B. B. Baldaniya, " Synthesis and Characterizations of (2Z)-ethyl-2-(Aryl)-3,5,8,8a-tetrahydro-5-(4-methoxyphenyl)-7-methyl-3-oxo-2H-oxazolo[3,2-a]pyrimidine-6-carboxylate as Biological Active Agents, International Journal of Scientific Research in Science and Technology(IJSRST), Online ISSN : 2395-602X, Print ISSN : 2395-6011, Volume 3, Issue 3, pp.362-365, March-April-2017.