Synthesis and Characterizations of (2Z)-ethyl-2-(Aryl)-3,5,8,8a-tetrahydro-5-(4-methoxyphenyl)-7-methyl-3-oxo-2H-oxazolo[3,2-a]pyrimidine-6-carboxylate as Biological Active Agents

Authors(2) :-J. S. Makwana, Dr. B. B. Baldaniya

Pyrimidine plays a significant role among other heterocycles. Pyrimidine nucleus was synthesized by Biginelli reaction. The purpose of this study was to synthesize several oxazolo derivative compounds (1-13) and evaluate them for their antibacterial activity. The structures of all title compounds have been confirmed on the basis of their analytical, IR spectral data. The title compounds have been tested for antibacterial and antifungal activities against different strains of bacteria.

Authors and Affiliations

J. S. Makwana
Department of Chemistry, M. G. Science institute, Navarangpura, Ahmedabad, Gujarat, India
Dr. B. B. Baldaniya
Department of Chemistry, M. G. Science institute, Navarangpura, Ahmedabad, Gujarat, India

Oxazolo Pyrimidine, Antibacterial activity, antifungal activities, Biginelli reaction.

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Publication Details

Published in : Volume 3 | Issue 3 | March-April 2017
Date of Publication : 2017-04-30
License:  This work is licensed under a Creative Commons Attribution 4.0 International License.
Page(s) : 362-365
Manuscript Number : IJSRST1733124
Publisher : Technoscience Academy

Print ISSN : 2395-6011, Online ISSN : 2395-602X

Cite This Article :

J. S. Makwana, Dr. B. B. Baldaniya, " Synthesis and Characterizations of (2Z)-ethyl-2-(Aryl)-3,5,8,8a-tetrahydro-5-(4-methoxyphenyl)-7-methyl-3-oxo-2H-oxazolo[3,2-a]pyrimidine-6-carboxylate as Biological Active Agents, International Journal of Scientific Research in Science and Technology(IJSRST), Print ISSN : 2395-6011, Online ISSN : 2395-602X, Volume 3, Issue 3, pp.362-365, March-April-2017. Available at doi : 10.32628/IJSRST1733124
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