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An Efficient and Green Synthesis of 1, 5-Benzodiazepines

Authors(4) :-Kishan P. Haval, Bhaurao P. Sathe, Pramod S. Phatak, Radhakrishnan M. Tigote

An efficient and green synthesis of 1, 5-Benzodiazepines is reported under neutral conditions. The ammonium chloride catalyzed condensation of o-phenylenediamine with several ketones in methanol at room temperature furnished corresponding 1, 5-benzodiazopines.
Kishan P. Haval, Bhaurao P. Sathe, Pramod S. Phatak, Radhakrishnan M. Tigote
1, 5-Benzodiazepines, O-Phenylenediamine, Ketones, Green Chemistry, Neutral Conditions.
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Publication Details
  Published in : Volume 3 | Issue 9 | November-December 2017
  Date of Publication : 2017-12-15
License:  This work is licensed under a Creative Commons Attribution 4.0 International License.
Page(s) : 95-99
Manuscript Number : IJSRST173919
Publisher : Technoscience Academy
PRINT ISSN : 2395-6011
ONLINE ISSN : 2395-602X
Cite This Article :
Kishan P. Haval, Bhaurao P. Sathe, Pramod S. Phatak, Radhakrishnan M. Tigote, "An Efficient and Green Synthesis of 1, 5-Benzodiazepines", International Journal of Scientific Research in Science and Technology(IJSRST), Print ISSN : 2395-6011, Online ISSN : 2395-602X, Volume 3, Issue 9, pp.95-99, November-December-2017
URL : http://ijsrst.com/IJSRST173919