Recent Advances in the Synthesis of Benzothiazoles : A Review

Authors

  • Rameshwar R. Magar  Department of Chemistry, Sant Dnyaneshwar Mahavidyalaya Soegaon, Dist. Aurangabad, Maharashtra, India

DOI:

https://doi.org/10.32628/IJSRST2310129

Keywords:

Benzothiazole, Pharmacological activities, Synthesis.

Abstract

Benzothiazoles are important heterocyclic compound because of their wide range of biological and pharmacological activity. In literature, it is reported that Benzothiazoles and its derivatives possess numerous pharmacological activities like antitumor, anticonvulsant, antimicrobial, antioxidant, antitubercular, antimalarial, antifungal, anti-inflammatory and antidiabetic activities. In recent year several methods have been developed for the synthesis of Benzothiazole derivatives due to their importance in bioorganic and medicinal chemistry. The present review focuses on systematic literature report of various synthetic procedures of Benzothiazoles derivatives using different strategies from the period 2010 to 2021.

References

  1. I. Hutchinson, T.D. Bradshaw, C.S. Matthews, M.F.G. Stevens, A.D. Westwell, Bioorg. Med. Chem. Lett., 13, (2003), 471-474.
  2. S.T. Huang, I. J. Hsei, C. Chen, Bioorg. Med. Chem., 14, (2006), 6106-6119.
  3. R.J. Alaimo, S.S. Pelosi, R. Freedman, J. Pharm. Sci., 67, (1978), 281-282.
  4. A.D. Borthwick, D.E. Davies, P.F. Ertl, A.M. Exall, T.M. Haley, G.J. Hart, D.L. Jackson, N.R. Parry, A. Patikis, N. Trivedi, G.G. Weingarten, J.M. Woolven, J. Med. Chem., 46, (2003), 4428-4449.
  5. G. Sreenivasa, E. Jayachandran, B. Shivakumar, K. Jayaraj and M. Kumar Vijay, Arch. Pharm. Sci. Res., 1, (2009), 150-157.
  6. X. Su, N. Vicker, D. Ganeshapillai, A. Smith, A. Purohit, M. J. Reed and B. V. Potter, Mol. Cell. Endocrinol., 248, (2006), 214-217.
  7. J. Neres, M. L. Brewer, L. Ratier, H. Botti, A. Buschiazzo, P. N. Edwards, P. N. Mortenson, M. H. Charlton, P. M. Alzari and A. C. Frasch, Bioorg. Med. Chem. Lett., 19, (2009), 589-596.
  8. D. Cressier, C. Prouillac, P. Hernandez, C. Amourette, M. Diserbo, C. Lion and G. Rima, Bioorg. Med. Chem., 17, (2009), 5275-5284.
  9. A. Benazzouz, T. Boraud, P. Dubedat, A. Boireau, J.-M. Stutzmann and C. Gross, Eur. J. Pharmacol., 284, (1995), 299-307.
  10. P. Jimonet, F. Audiau, M. Barreau, J.-C. Blanchard, A. Boireau, Y. Bour, M.-A. Coleno, A. Doble, G. Doerflinger and C. Do Huu, J. Med. Chem., 42, (1999), 2828-2843.
  11. I. Hutchinson, S. A. Jennings, B. R. Vishnuvajjala, A. D. Westwell and M. F. Stevens, J. Med. Chem., 45, (2002), 744-747.
  12. S. Nadeem, A. Rana, S. A. Khan, S. E. Haque, M. S. Alam and W. Ahsana, Acta Chim. Slov., 56, (2009), 462-469.
  13. R. Danzeisen, B. Schwalenstoecker, F. Gillardon, E. Buerger, V. Krzykalla, K. Klinder, L. Schild, B. Hengerer, A. C. Ludolph and C. Dorner-Ciossek, J. Pharmacol. Exp. Ther., 316, (2006), 189-199.
  14. B. Gurupadayya, Y. Manohara and M. Gopal, Indian J. Heterocycl. Chem., 15, (2006), 113-116.
  15. B. Rajeeva, N. Srinivasulu and S. Shantakumar, J. Chem., 6, (2009), 775-779.
  16. S.C. Debnath, D.K. Basu, J. Appl. Polym. Sci. 52, (1994), 597-603.
  17. C.P. Ye, N.G. Wang, H.Q. Jia, X.J. Xu, Chin. J. Appl. Chem., 19, (2002), 1008-1010.
  18. A. Heynderickx, R. Guglielmetti, R. Dubest, J. Aubard, A. Samat, Synthesis, (2003), 1112-1116.
  19. B.C. Lee, J.S. Kim, B.S. Kim, J.Y. Son, S.K. Hong, H.S. Park, B.S. Moon, J.H. Jung, J.M. Jeong, S.E. Kim, Bioorg. Med. Chem., 19, (2011), 2980-2990.
  20. A. A. Weekes, M. C. Dix, M. C. Bagley, A. D. Westwell, Synth. Commun., 40, (2010), 3027-3032.
  21. B. S. Londhe, U. R. Pratap, J. R. Mali, R. A. Mane, Bull. Korean Chem. Soc., 31, (2010), 2329-2332.
  22. S. V. Nalage, S. V. Bhosale, D. S. Bhosale, W. N. Jadhav, Chin. Chem. Lett., 21, (2010), 790-793.
  23. B. Maleki, H. Salehabadi, M. K. Moghaddan, Acta Chim. Slov., 57, (2010), 741-745.
  24. V. Hojat, G. V. Ramin, F.Alireza, O. Turan, Chin. J. Chem., 28, (2010), 2249-2254.
  25. S. S. Katkar, P. H. Mohite, L. S. Gadekar,K. N. Vidhate, M. K. Lande, Chin. Chem. Lett., 21 (2010) 421-425.
  26. T. G. Deligeorgiev, S. Kaloyanova, A. Vasilev, J. J. Vaquero, Phosphorus, Sulfur, and Silicon, 185, (2010) 2292–2302.
  27. S. Sadjadi, H. Sepehrian, Ultrason. Sonochem., 18, (2011), 480-483.
  28. Y. Yuan, S. Guo, Synth. Commun., 41, (2011), 2169-2177.
  29. P. Bandyopadhyay, M. Sathe, G. K. Prasad, P. Sharma, M. P. Kaushik, J. Mol. Catal.A Chem., 341, (2011), 77-82.
  30. A. Shokrolahi, A. Zali, M. Mahdavi, Phosphorous, Sulphur and Silicon, 187, (2012), 535-543.
  31. A. Rostami and A. Yari, J. IRAN CHEM SOC., 9, (2012), 489-493.
  32. K. U. Sadek, R. A. Mekheimer, A. M. A. Hameed, F. Elnahas, M. H. Elnagdi, Molecule, 17, (2012), 6011-6019.
  33. L. Zhang, J. Xia, Y. Zhou, H. Wang, S. Wang, Synth. Commun., 42, (2012), 328-336.
  34. H. Eshghi, M. Rahimizadeh, A. Shiri, P. Sedaghat, Bull. Korean Chem. Soc., 33, (2012), 515-518.
  35. G. F. Chen, L. Y. Zhang, H. M. Jia, B. H. Chen, J. T. Li, S. X. Wang, G. Y. Bai. Res. Chem. Intermed., 39, (2013), 2077-2086.
  36. G. F. Chen, H. M. Jia, L. Y. Zhang, B. H. Chen, J. T. Li, Ultrason. Sonochem., 20, (2013), 627-632
  37. M. Ghashang, Res. Chem. Intermed., 40, (2014), 1669-1674
  38. G. F. Chen, N. Xiao, J. S. Yang, H. Y. Li, B. H. Chen, L. F. Han, Res. Chem. Intermed., 41, (2015), 5159-5166.
  39. A. Amoozadeh, R. A. Azadeh, S. Rahmani, M Salehi, M. Kubicki, G. Dutkiewicz, Phosphorous, Sulphur and Silicon and related element, 190, (2015), 1874-1883.
  40. C. H. Gill, M. D. Nikam, P. S. Mahajan, A. V. Chate, S. K. Dabhade, P. V. Badadhe, Res. Chem. Intermed, 41, (2015), 7509-7516.
  41. Z. Y. Yu, Q. S. Fang, J. Zhou, Z. B. Song, Res. Chem. Intermed., 42, (2016), 2035-2045.
  42. A. V. Borhade, B. K. Uphade, A. G. Gadhave, Res. Chem. Intermed., 42, (2016), 6301-6311.
  43. B. F. Mirjalili, A. Bamoniri, M. A. Mirhoseini, Iran. J. Catal., 6, (2016), 23-27.
  44. K. D. Dhawale, A. P. Ingale, S. V. Shinde, N. M. Thorat, L. R. Patil, Synth. Commun., 51, (2021), 1588-1601.
  45. S. P. Gadekar, M. K. Lande, Res. Chem. Intermed., 47, (2021), 1253-1267.

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Published

2023-02-28

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Research Articles

How to Cite

[1]
Rameshwar R. Magar "Recent Advances in the Synthesis of Benzothiazoles : A Review " International Journal of Scientific Research in Science and Technology(IJSRST), Online ISSN : 2395-602X, Print ISSN : 2395-6011,Volume 10, Issue 1, pp.282-291, January-February-2023. Available at doi : https://doi.org/10.32628/IJSRST2310129